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   CAS NO.    Products Name
   1086062-66-9 GSK 2126458  more...
   GSK2126458 is a highly potent PI3K and mTOR inhibitor with an app Ki of 19 pM for PI3K. In vivo, GSK2126458 showed anti-tumor activity in both pharmacodynamic and tumor growth efficacy ...
   1201438-56-3 IPI-145  more...
   IPI-145 is an orally bioavailable, highly selective and potent small molecule inhibitor of the delta and gamma isoforms of phosphoinositide-3 kinase (PI3K) with potential immunomodulati...
   371242-69-2 IC-87114  more...
   IC-87114 is the first isoform-selective PI3K inhibitor. This quinazolinone purine inhibits p110δ(IC50=0.13µM) at mid-nanomolar concentrations and shows 100–1000-fold selectivity o...
   154447-36-6 LY 294002  more...
   LY294002 inactivates Akt/PKB, consequently inhibiting cell proliferation and inducing apoptosis. LY294002 demonstrates a remarkable growth-inhibitory and apoptosis-inducing effect in th...
   1245537-68-1 NVP-BGT226  more...
   NVP-BGT226 has entered phase I/II clinical trials for the treatment of advanced solid tumors (including breast cancer)....
   944396-07-0 NVP-BKM-120  more...
   BKM120 (NVP-BKM120) is a bioavailable specific oral pan-class I phosphatidylinositol 3-kinase (PI3K) kinase inhibitor. BKM120 inhibits tumor proliferation and survival by blocking the p...
   915019-65-7 NVP-BEZ 235  more...
   BEZ235 (NVP-BEZ235) inhibits PI3K and mTOR kinase activity by binding to the ATP-binding cleft of these enzymes. The phosphatidylinositol 3-kinase (PI3K)/Akt/mammalian target of rapamyc...
   677338-12-4 PIK-90  more...
   PIK-90 is a potent and cell permeable PI3K inhibitor, with IC50 values (nM) of 11, 350, 18, and 58 for p110 α, β, γ and δ isoforms, low mTOR activity. Besides Val882 H-binding, PIK-90 u...
   1197160-78-3 PKI-587  more...
   PKI-587 is a highly potent dual PI3K/mTOR kinase inhibitor with IC50 of 0.4 nM and <0.1 μM for PI3K-α and mTOR, respectively. Intravenous administration of PKI-587 exhibits excellent an...
   157716-52-4 Perifosine  more...
   Biological Activity of Perifosine: A p.o.-bioavailable ALK(Alkylphospholipids),inhibits Akt activation. Targeting cellular membranes, perifosine modulates membrane permeability, membra...

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